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Metronidazole

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Ibicuruzwa birambuye

Ibicuruzwa

Ibicuruzwa birambuye

CAS: 443-48-1

1.Metronidazole ni antibiyotike ya nitroimidazole, izwi kandi nka methotrexate, metronidazole, metronidazole, metronidazole, methotrexate, mikorobe ya anaerobic igira ingaruka zo kwica, igabanuka mu mubiri w'umuntu iyo metabolite yakozwe nayo igira ingaruka za bagiteri zirwanya anaerobic. synthesis ya acide deoxyribonucleic ya bagiteri, bityo ikabangamira imikurire ya bagiteri, imyororokere, kandi amaherezo igatera urupfu rwa bagiteri, bagiteri zirwanya anaerobic Pu zirimo: Bacteroides fragilis, Clostridium (bitewe na bagiteri zirwanya anaerobic zirimo: Bacteroides fragilis, Clostridium perfringens ( yitiriwe kubera impera zikarishye za bagiteri), Bacillus tetani, Streptococcus pepticus, Streptococcus pepticus, na JaChemicalbook flagellate. Byabanje gukoreshwa mu kuvura trichomoniasis yo mu nda ibyara bifite akamaro gakomeye mu mavuriro. Nyuma byaje kugaragara ko metronidazole ishobora no kwica bagiteri ya anaerobic. gutera indwara zo mu kanwa, kandi mu 1978 byamenyekanye na World Umuryango w’ubuzima nkumuti ukomeye urwanya indwara ya anaerobic kandi ukoreshwa cyane mukurinda no kuvura indwara zo mu kanwa.Ikoreshwa kandi mubitaro mugukumira no kuvura indwara zubuhumekero, gastrointestinal, abdominal na pelvic infection ziterwa na bagiteri ya anaerobic, indwara zuruhu nudukoko tworoshye, indwara zamagufwa n ingingo zifatanije, karite, sepsis nubwonko.

2.Uburyo bwibikorwa ni mukubuza redox reaction ya amoeba protozoa, kugirango urunigi rwa azote ya protozoa rucike n'ingaruka.Mu isuzuma rya vitro ryerekana ko kuri concentration ya 1 ~ 2mg / L, ihinduka ryimiterere ya ameba ya tissue ya Chemical Book rishobora kubaho mumasaha 6 ~ 20, kandi bose barashobora kwicwa mumasaha 24.

3. Ifu yera cyangwa umuhondo kristu cyangwa ifu ya kristaline;impumuro nziza, isharira kandi umunyu muke.Gushonga buhoro muri Ethanol, gushonga gake mumazi cyangwa chloroform, gushonga gato muri ether.Methyl Chemical Book nitrazole ni azote irimo ibinyabuzima bya heterocyclic hamwe na alkaline hamwe no gukomera kwamazi.Ukurikije ihame ryo guteganya, metronidazole ikorwa mu munyu wa potasiyumu ya fosifate, kandi amazi yiyongera, ashobora gukoreshwa nk'umuti wo gutera inshinge.

Gusaba

1.Yakoreshejwe mu kuvura trichomoniasis kuva 1959 no muri amibe yo munda yo munda no hanze kuva 1970, hamwe nubushobozi buhanitse, uburozi buke no gukoreshwa cyane.Ifite ingaruka za mutagenic na teratogenic mubushakashatsi bwinyamaswa.
2.Ingaruka zikomeye za antibacterial kurwanya bagiteri nyinshi za anaerobic
3.Ku kuvura amibeya, trichomoniasis n'indwara ya anaerobic

 


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